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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T10026 | Tachykinin angatonist 1 | Tachykinin antagonist 1 | Others |
Tachykinin antagonist 1 is an antagonist of neurokinin receptors. | |||
T14524 | Befetupitant | Ro67-5930 | Neurokinin receptor |
Befetupitant (Ro67-5930) is a potent and selective tachykinin 1 receptor (NK1R) antagonist for the study of corneal neovascularization. | |||
T69140 | Burapitant | SSR 240600 | Neurokinin receptor |
Burapitant (SSR 240600) is a novel non-peptide tachykinin neurokinin 1 (NK) receptor antagonist with anti-coke oven and antidepressant activity. | |||
T12000 | MEN11467 | Neurokinin receptor | |
MEN11467 is a novel, orally available, potent and selective peptidomimetic tachykinin NK 1 receptor antagonist for the study of acute colon cancer. | |||
T28917 | TAK-637 | TAK 637 | |
TAK-637 is a tachykinin 1 (NK1) receptor antagonist. | |||
T28706 | SCH 206272 | SCH206272,SCH-206272 | |
SCH 206272 is a potent, orally active antagonist of tachykinin NK(1), NK(2), and NK(3) receptor. | |||
T69184 | Figopitant | ||
Figopitant is a tachykinin neurokinin-1 antagonist. | |||
T83496 | [D-Pro4,D-Trp7,9,10] Substance P (4-11) | ||
[D-Pro4,D-Trp7,9,10] Substance P (4-11) serves as a potent antagonist of the tachykinin family of neuropeptides [1]. | |||
T29185 | YM44781 | YM 44781,YM-44781 | |
YM44781 is a non-peptide tachykinin receptor antagonist. YM44781 exhibits high binding affinities at NK(1) (pK(i) = 9.09 +/- 0.02) and NK(2) (pK(i) = 9.94 +/- 0.03) receptors, respectively. | |||
T75879 | Men 10376 TFA | ||
Men 10376 TFA is a selective antagonist of the tachykinin NK-2 receptor, displaying a K i value of 4.4 μM specifically for the NK-2 receptor in rat small intestine [1]. | |||
T29186 | YM49598 | YM-49598,YM 49598 | |
YM49598 is a tachykinin receptor antagonist. YM49598 exhibited high binding affinities at NK(1) (pK(i) = 9.09 +/- 0.02) and NK(2) (pK(i) = 9.94 +/- 0.03) receptors, respectively. YM49598 was almost inactive but produced ... | |||
T76405 | [D-Trp2,7,9] Substance P | ||
[D-Trp2,7,9] Substance P is a tachykinin (Neurokinin Receptor) antagonist that exhibits inhibitory affinities (K_i values) of 1 μM for NK-1, 1.3 μM for NK-2, and approximately 9 μM for NK-3 receptors [1]. |